| Round | Overall | Player |
|---|---|---|
| 1 | 4th | SP Mark Prior ChN |
| 2 | 21st | SS Edgar Renteria StL |
| 3 | 28th | OF Vernon Wells Tor |
| 4 | 45th | SP Barry Zito Oak |
| 5 | 52nd | OF Brian S. Giles SD |
| 6 | 69th | SP Johan Santana Min |
| 7 | 76th | OF Miguel Cabrera Fla |
| 8 | 93rd | 3B Aramis Ramirez ChN |
| 9 | 100th | SS Mike Young Tex |
| 10 | 117th | 1B Paul Konerko ChA |
| 11 | 124th | OF Corey Patterson ChN |
| 12 | 141st | SP Rich Harden Oak |
| 13 | 148th | C Paul Lo Duca Fla |
| 14 | 165th | C Ramon Hernandez SD |
| 15 | 172nd | SP Jake Peavy SD |
| 16 | 189th | SP Kelvim Escobar Ana |
| 17 | 196th | SP Rafael Soriano Sea |
| 18 | 213th | RP Ugueth Urbina Det |
| 19 | 220th | OF Jacque Jones Min |
| 20 | 237th | 3B Adrian Beltre LA |
| 21 | 244th | SP Adam Eaton SD |
| 22 | 261st | RP Shingo Takatsu ChA |
| 23 | 268th | SP Ryan Wagner Cin |
| 24 | 285th | OF Luis Matos Bal |
| 25 | 292nd | SP Wilson Alvarez LA |
| 26 | 309th | SP A.J. Burnett Fla |
| 27 | 316th | OF Alexis Rios Tor |
| 28 | 333rd | 1B Lyle Overbay Mil |
| 29 | 340th | SP Jon Lieber NYA |